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Upacicalcet sodium 

Cat. No.: HY-109106A Purity: ≥98.0%
Handling Instructions

Upacicalcet sodium is an intravenous calcimimetic agent. Upacicalcet suppresses excessive parathyroid hormone (PTH) secretion, thereby lowering blood PTH levels, by acting directly on parathyroid cell membrane calcium-sensing receptors. Upacicalcet can be used for researching the disease of secondary hyperparathyroidism (SHPT).

For research use only. We do not sell to patients.

Upacicalcet sodium Chemical Structure

Upacicalcet sodium Chemical Structure

CAS No. : 2052969-18-1

Size Price Stock Quantity
5 mg USD 752 In-stock
Estimated Time of Arrival: December 31
10 mg USD 1200 In-stock
Estimated Time of Arrival: December 31
25 mg USD 2640 In-stock
Estimated Time of Arrival: December 31
50 mg USD 4304 In-stock
Estimated Time of Arrival: December 31
100 mg USD 6880 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

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Description

Upacicalcet sodium is an intravenous calcimimetic agent. Upacicalcet suppresses excessive parathyroid hormone (PTH) secretion, thereby lowering blood PTH levels, by acting directly on parathyroid cell membrane calcium-sensing receptors. Upacicalcet can be used for researching the disease of secondary hyperparathyroidism (SHPT)[1].

IC50 & Target

calcium-sensing receptors[1]

Molecular Weight

373.75

Formula

C11H13ClN3NaO6S

CAS No.
SMILES

O=C(NC[[email protected]](N)C(O[Na])=O)NC1=CC(S(=O)(O)=O)=CC(Cl)=C1C

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

-20°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (267.56 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.6756 mL 13.3779 mL 26.7559 mL
5 mM 0.5351 mL 2.6756 mL 5.3512 mL
10 mM 0.2676 mL 1.3378 mL 2.6756 mL
*Please refer to the solubility information to select the appropriate solvent.
Purity & Documentation

Purity: ≥98.0%

References
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Product Name:
Upacicalcet sodium
Cat. No.:
HY-109106A
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