VU6008677
VU6008677 is a positive allosteric modulator (PAM) for M4, with EC50 of 120 nM for hM4. VU6008677 inhibits cytochrome P450, exhibits good pharmacokinetic characteristics in rats.
For research use only. We do not sell to patients.
- CAS No.: 2170550-99-7
- Formula: C14H13ClN4O
- Molecular Weight:288.73
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
EC50: 120 nM (hM4)
Chemical Information
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CAS No. 2170550-99-7
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Molecular Weight 288.73
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Formula C14H13ClN4O
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SMILES
CC1=C(Cl)C(C)=NC2=C1C3=C(C(NC4CC4)=NC=N3)O2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)