1. GPCR/G Protein
  2. LPL Receptor

BMS-986020 (Synonyms: AM152)

Cat. No.: HY-100619 Purity: 98.02%
Handling Instructions

BMS-986020 is an LPA1 antagonist.

For research use only. We do not sell to patients.

BMS-986020 Chemical Structure

BMS-986020 Chemical Structure

CAS No. : 1257213-50-5

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 127 In-stock
Estimated Time of Arrival: December 31
1 mg USD 80 In-stock
Estimated Time of Arrival: December 31
5 mg USD 120 In-stock
Estimated Time of Arrival: December 31
10 mg USD 170 In-stock
Estimated Time of Arrival: December 31
50 mg USD 450 In-stock
Estimated Time of Arrival: December 31
100 mg USD 750 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

BMS-986020 is an LPA1 antagonist. target: LPA1 BMS-986020 is in Phase 2 clinical development for treating idiopathic pulmonary fibrosis. BMS-986020 selectively inhibits the LPA receptor, which is involved in binding of the signaling molecule lysophosphatidic acid, which in turn is involved in a host of diverse biological functions, such as cell proliferation, platelet aggregation, smooth muscle contraction and others.

Clinical Trial
Solvent & Solubility
In Vitro: 

DMSO : ≥ 64 mg/mL (132.63 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.0724 mL 10.3621 mL 20.7241 mL
5 mM 0.4145 mL 2.0724 mL 4.1448 mL
10 mM 0.2072 mL 1.0362 mL 2.0724 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

482.53

Formula

C₂₉H₂₆N₂O₅

CAS No.

1257213-50-5

SMILES

O=C(C1(C2=CC=C(C3=CC=C(C4=C(NC(O[[email protected]@H](C5=CC=CC=C5)C)=O)C(C)=NO4)C=C3)C=C2)CC1)O

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Inquiry Online

Your information is safe with us. * Required Fields.

Product name

 

Salutation

Applicant name *

 

Email address *

Phone number *

 

Organization name *

Country or Region *

 

Requested quantity *

Remarks

Bulk Inquiry

Inquiry Information

Product Name:
BMS-986020
Cat. No.:
HY-100619
Quantity:

BMS-986020

Cat. No.: HY-100619