1. Epigenetics
  2. Histone Acetyltransferase
  3. Histone Acetyltransferase Inhibitor II

Histone Acetyltransferase Inhibitor II 

Cat. No.: HY-100734 Purity: 99.11%
Handling Instructions

Histone Acetyltransferase Inhibitor II is a potent and cell permeable p300 inhibitor, with an IC50 of 5 µM; Histone Acetyltransferase Inhibitor II can be used in cancer research.

For research use only. We do not sell to patients.

Histone Acetyltransferase Inhibitor II Chemical Structure

Histone Acetyltransferase Inhibitor II Chemical Structure

CAS No. : 932749-62-7

Size Price Stock Quantity
Free Sample (0.5-1 mg)   Apply now  
10 mM * 1 mL in DMSO USD 92 In-stock
Estimated Time of Arrival: December 31
5 mg USD 84 In-stock
Estimated Time of Arrival: December 31
10 mg USD 132 In-stock
Estimated Time of Arrival: December 31
25 mg USD 264 In-stock
Estimated Time of Arrival: December 31
50 mg USD 456 In-stock
Estimated Time of Arrival: December 31
100 mg USD 780 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

Based on 1 publication(s) in Google Scholar

Top Publications Citing Use of Products
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  • Purity & Documentation

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Description

Histone Acetyltransferase Inhibitor II is a potent and cell permeable p300 inhibitor, with an IC50 of 5 µM; Histone Acetyltransferase Inhibitor II can be used in cancer research.

IC50 & Target

IC50:5 µM (p300)[1]

Molecular Weight

464.15

Formula

C₂₀H₁₆Br₂O₃

CAS No.

932749-62-7

SMILES

O=C1/C(CCC/C1=C\C2=CC=C(O)C(Br)=C2)=C/C3=CC=C(O)C(Br)=C3

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : ≥ 30 mg/mL (64.63 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.1545 mL 10.7724 mL 21.5448 mL
5 mM 0.4309 mL 2.1545 mL 4.3090 mL
10 mM 0.2154 mL 1.0772 mL 2.1545 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.5 mg/mL (5.39 mM); Clear solution

*All of the co-solvents are provided by MCE.
References

Purity: 99.11%

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Keywords:

Histone Acetyltransferase Inhibitor IIHistone AcetyltransferaseHATsHATInhibitorinhibitorinhibit

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Product name:
Histone Acetyltransferase Inhibitor II
Cat. No.:
HY-100734
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