Altanserin hydrochloride
Altanserin is a 5-hydroxytryptamine (5-HT2A ) selective radioligand. Altanserin delivers human serotonin. Altanserin can be used to study the biochemical and cellular mechanisms of vulnerability to extracellular 5-HT increase .
For research use only. We do not sell to patients.
- CAS No.: 1135280-78-2
- Formula: C22H23ClFN3O2S
- Molecular Weight:447.95
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All 5-HT Receptor Isoforms
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Biological Activity
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5-HT2A Receptor |
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| U2OS | IC50 |
1.51 nM
Compound: Altanserin
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Antagonist activity at recombinant human 5-HT2A expressed in human U2OS cells by pathhunter beta-arrestin assay
Antagonist activity at recombinant human 5-HT2A expressed in human U2OS cells by pathhunter beta-arrestin assay
|
[PMID: 32631554] |
Chemical Information
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CAS No. 1135280-78-2
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Molecular Weight 447.95
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Formula C22H23ClFN3O2S
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SMILES
O=C1N(CCN2CCC(C(C3=CC=C(F)C=C3)=O)CC2)C(NC4=C1C=CC=C4)=S.Cl
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)