BRD4-IN-10
BRD4-IN-10 (Compound 31) is a selective BRD4 inhibitor with an IC50 of 13.5 nM. BRD4-IN-10 can exert anti-inflammatory and anti-fibrotic effects. BRD4-IN-10 also has good metabolic stability, pharmacokinetic properties and safety. BRD4-IN-10 can be used in the research of renal fibrosis diseases.
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- CAS. Nr.: 3051852-76-4
- Formel: C24H30N8O3
- Molecular Weight:478.55
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biologische Aktivität
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BRD4 (BD1) 13.5 nM (IC50) |
Chemical Information
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CAS. Nr. 3051852-76-4
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Molecular Weight 478.55
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Formel C24H30N8O3
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SMILES
O=C1NC(C2(CCN(C3=NC(NC4=CC(N(C(C)C)[C@H](C)C(N5C)=O)=C5C=C4)=NC=C3)CC2)N1)=O
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)