KSK68
KSK68 is a high-affinity dual sigma-1 and histamine H3 receptor antagonist, with Kis of 7.7, 3.6, 22.4 nM for H3 receptor, sigma-1, sigma-2 receptor respectively. KSK68 has negligible affinity at the other histamine receptor subtypes. KSK68 can be used for research of nociceptive and neuropathic pain.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- CAS. Nr.: 2566715-91-9
- Formel: C23H28N2O2
- Molecular Weight:364.48
-
Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Alle Sigma Receptor Isoform-spezifische Produkte anzeigen
MoreAlle Histamine Receptor Isoform-spezifische Produkte anzeigen
More
Biologische Aktivität
7.7 nM, 3.6 nM、22.4 nM (H3 receptor, sigma-1, sigma-2 receptor)[1]
Chemical Information
-
CAS. Nr. 2566715-91-9
-
Molecular Weight 364.48
-
Formel C23H28N2O2
-
SMILES
O=C(C1CC1)C2=CC=C(OCCCN3CCC(C4=CC=NC=C4)CC3)C=C2
-
Versand
Room temperature in continental US; may vary elsewhere.
-
Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)