SR 1824
SR 1824 is a non-agonist PPARγ ligand that blocks Cdk5-mediated phosphorylation. SR 1824 has anti-diabetic effects.
For research use only. We do not sell to patients.
- CAS No.: 1338259-06-5
- Formula: C33H29BrN2O3
- Molecular Weight:581.50
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| HEK-293T | EC50 |
516 nM
Compound: 37
|
Transactivation of human PPARgamma in HEK293T cells after 18 hrs by luciferase reporter gene assay
Transactivation of human PPARgamma in HEK293T cells after 18 hrs by luciferase reporter gene assay
|
[PMID: 26396687] |
Chemical Information
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CAS No. 1338259-06-5
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Molecular Weight 581.50
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Formula C33H29BrN2O3
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SMILES
O=C(C1=CC=CC=C1C2=CC=C(CN3C(C)=C(C)C4=C3C=CC(C(N[C@H](C5=CC=C(Br)C=C5)C)=O)=C4)C=C2)O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)