1. Metabolic Enzyme/Protease
  2. Phosphodiesterase (PDE)
  3. Autotaxin-IN-3

Autotaxin-IN-3 

Cat. No.: HY-135053
Handling Instructions

Autotaxin-IN-3 is a Autotaxin(ATX) inhibitor with an IC50 of 2.4 nM, compound 33, sourced from patent WO2018212534A1.

For research use only. We do not sell to patients.

Autotaxin-IN-3 Chemical Structure

Autotaxin-IN-3 Chemical Structure

CAS No. : 2156655-68-2

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 341 In-stock
Estimated Time of Arrival: December 31
5 mg USD 350 In-stock
Estimated Time of Arrival: December 31
10 mg USD 550 In-stock
Estimated Time of Arrival: December 31
50 mg USD 1650 In-stock
Estimated Time of Arrival: December 31
100 mg USD 2250 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

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Based on 1 publication(s) in Google Scholar

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Description

Autotaxin-IN-3 is a Autotaxin(ATX) inhibitor with an IC50 of 2.4 nM, compound 33, sourced from patent WO2018212534A1[1].

IC50 & Target[1]

Autotaxin

2.4 nM (IC50)

In Vitro

Autotaxin is an enzyme which is responsible for the increase in lysophosphatidic acid in ascites and plasma, and it is a secretory enzyme important for converting lysophosphatidylchloine (LPC) into lysophosphatidic acid (LPA) as a bioactive signaling molecule[1].

Molecular Weight

443.46

Formula

C₂₂H₂₁N₉O₂

CAS No.

2156655-68-2

SMILES

O=C(N1CCC(N=NN2)=C2C1)CC3=NN=C(C4=CN=C(NC5CC6=C(C=CC=C6)C5)N=C4)O3

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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Keywords:

Autotaxin-IN-3Phosphodiesterase (PDE)IdiopathicPulmonaryFibrosisIPF,Inhibitorinhibitorinhibit

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