JYL 1511
JYL 1511 is a partial agonist of vanilloid receptor VR1.
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- CAS No.: 623166-14-3
- Formule: C21H29N3O3S2
- Masse moléculaire:435.60
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| CHO | EC50 |
32.4 nM
Compound: 3
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Agonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assay
Agonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assay
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[PMID: 18406014] |
JYL 1511 inhibits [3H]Resiniferatoxin binding to rat VR1 with a Ki of 50.4 nM[1].
JYL 1511 inhibits Capsaicin induction of 45Ca2+ uptake in CHO cells overexpressing rat VR1 (IC50: 3.4 nM)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 623166-14-3
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Masse moléculaire 435.60
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Formule C21H29N3O3S2
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SMILES
CS(=O)(NC1=CC=C(C=C1OC)CNC(NCC2=CC=C(C=C2)C(C)(C)C)=S)=O
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
JYL 1511 Related Classifications
HY-118299 Related Classifications
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