SYAF080
SYAF080 is a human A₂B adenosine receptor (hA₂B AdoR) antagonist with a Ki of 23.6 nM and a KB of 25.2 nM. SYAF080no relevant inhibition of human CYP450 cytochromes. SYAF080 can be used for the research of inflammation, metabolic and cardiovascular disease.
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- CAS No.: 352692-70-7
- Formule: C12H14N2O3S
- Masse moléculaire:266.32
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
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Activité biologique
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hA2B 23.6 nM (Ki) |
hA2B 25.2 nM (Kb) |
SYAF080 (Compound 21a) (10 µM) inhibits hA1, hA2A, hA2B and hA3 (Ki = 23.6 nM for hA2B; KB = 25.2 nM) and inhibits c-AMP production[1].
SYAF080 shows no relevant inhibition of human CYP450 cytochrome[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 352692-70-7
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Masse moléculaire 266.32
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Formule C12H14N2O3S
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SMILES
O=C(OCC)C1=C(NC(=O)NC1C2=CSC=C2)C
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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