1. Membrane Transporter/Ion Channel
    Neuronal Signaling
  2. Calcium Channel
  3. Carboxyamidotriazole

Carboxyamidotriazole (Synonyms: L-651582; CAI)

Cat. No.: HY-16126 Purity: ≥99.0%
Handling Instructions

Carboxyamidotriazole (L-651582) is a cytostatic inhibitor of nonvoltage-operated calcium channels and calcium channel-mediated signaling pathways. Carboxyamidotriazole shows anti-tumor, anti-inflammatory and antiangiogenic effects.

For research use only. We do not sell to patients.

Carboxyamidotriazole Chemical Structure

Carboxyamidotriazole Chemical Structure

CAS No. : 99519-84-3

Size Price Stock Quantity
Solution
10 mM * 1 mL in DMSO USD 280 In-stock
Estimated Time of Arrival: December 31
Solid + Solvent
10 mM * 1 mL
ready for reconstitution
USD 280 In-stock
Estimated Time of Arrival: December 31
Solid
1 mg USD 60 In-stock
Estimated Time of Arrival: December 31
5 mg   Get quote  
10 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

Other Forms of Carboxyamidotriazole:

Top Publications Citing Use of Products
  • Biological Activity

  • Purity & Documentation

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Description

Carboxyamidotriazole (L-651582) is a cytostatic inhibitor of nonvoltage-operated calcium channels and calcium channel-mediated signaling pathways. Carboxyamidotriazole shows anti-tumor, anti-inflammatory and antiangiogenic effects[1][2].

IC50 & Target

Calcium channel[1]

Clinical Trial
Molecular Weight

424.67

Formula

C17H12Cl3N5O2

CAS No.
Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (235.48 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.3548 mL 11.7738 mL 23.5477 mL
5 mM 0.4710 mL 2.3548 mL 4.7095 mL
10 mM 0.2355 mL 1.1774 mL 2.3548 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.5 mg/mL (5.89 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.5 mg/mL (5.89 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.5 mg/mL (5.89 mM); Clear solution

*All of the co-solvents are available by MCE.
References

Purity: ≥99.0%

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This equation is commonly abbreviated as: C1V1 = C2V2

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Product Name:
Carboxyamidotriazole
Cat. No.:
HY-16126
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