CCT369834
CCT369834 is an ATP-competitive HSET inhibitor with an IC50 of 39 nM. CCT369834 is a trans-cyclooctene-tagged probe. CCT369834 and HSET specifically co-localize on mitotic spindles. CCT369834 can be used for the research of cancer.
For research use only. We do not sell to patients.
- CAS No.: 2902671-78-5
- Formula: C38H49N7O7S
- Molecular Weight:747.90
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
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Biological Activity
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HSET 39 nM (IC50) |
CCT369834 inhibits recombinant full-length HSET (IC50 = 39 nM)[1].
CCT369834 (3 μM; 45 min) shows clear Cy5-labeled mitotic spindle signals in proTAME-treated DLD1 4N cells, which overlap with endogenous HSET signals[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2902671-78-5
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Molecular Weight 747.90
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Formula C38H49N7O7S
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SMILES
O=C(N[C@H](CC(NC1=NC(C)=C(S1)C(OCCC)=O)=O)CCCN(CC#CCNC(O[C@H]2CCC/C=C/CC2)=O)C)C3=CC=CC(C4=NOC(C)=N4)=C3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
CCT369834 Related Classifications
HY-180304 Related Classifications
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