1. Metabolic Enzyme/Protease
  2. Thrombin
  3. Dabigatran (ethyl ester)

Dabigatran (ethyl ester) 

Cat. No.: HY-17378 Purity: ≥98.0%
Handling Instructions

Dabigatran ethyl ester is an emerging oral anticoagulant which is a direct inhibitor of thrombin activity.

For research use only. We do not sell to patients.

Dabigatran (ethyl ester) Chemical Structure

Dabigatran (ethyl ester) Chemical Structure

CAS No. : 429658-95-7

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5 mg USD 96 In-stock
Estimated Time of Arrival: December 31
10 mg USD 156 In-stock
Estimated Time of Arrival: December 31
50 mg USD 528 In-stock
Estimated Time of Arrival: December 31
100 mg USD 840 In-stock
Estimated Time of Arrival: December 31
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Based on 1 publication(s) in Google Scholar

Other Forms of Dabigatran (ethyl ester):

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Description

Dabigatran ethyl ester is an emerging oral anticoagulant which is a direct inhibitor of thrombin activity. IC50 value: Target: thrombin Dabigatran provides a stable anticoagulation effect without any need to perform periodical laboratory controls. Of note, there is a growing amount of clinical evidence which shows its safety and efficacy. For these reasons, Dabigatran may suppose a revolution in oral anticoagulation. Dabigatran etexilate was rapidly converted to Dabigatran, with peak plasma dabigatran concentrations being attained after approximately 1.5 h; the bioavailability of Dabigatran after p.o. administration of Dabigatran etexilate was 7.2%.

Molecular Weight

499.56

Formula

C₂₇H₂₉N₇O₃

CAS No.

429658-95-7

SMILES

O=C(N(C1=NC=CC=C1)CCC(OCC)=O)C2=CC=C3C(N=C(N3C)CNC4=CC=C(C(N)=N)C=C4)=C2

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

H2O : 1 mg/mL (2.00 mM; ultrasonic and warming and heat to 80°C)

DMSO : 1 mg/mL (2.00 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.0018 mL 10.0088 mL 20.0176 mL
5 mM --- --- ---
10 mM --- --- ---
*Please refer to the solubility information to select the appropriate solvent.
References
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Keywords:

Dabigatran (ethyl ester)ThrombinInhibitorinhibitorinhibit

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Product Name:
Dabigatran (ethyl ester)
Cat. No.:
HY-17378
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