1. GPCR/G Protein
    Neuronal Signaling
  2. mAChR
  3. Emraclidine

Emraclidine 

Cat. No.: HY-132812
Handling Instructions

Emraclidine is a muscarinic M4 receptor positive allosteric modulator (WO2018002760, compound 11). Emraclidine can be used for the research of neurological diseases.

For research use only. We do not sell to patients.

Emraclidine Chemical Structure

Emraclidine Chemical Structure

CAS No. : 2170722-84-4

Size Price Stock
5 mg USD 450 Ask For Quote & Lead Time
10 mg USD 800 Ask For Quote & Lead Time
25 mg USD 1650 Ask For Quote & Lead Time
50 mg USD 2580 Ask For Quote & Lead Time
100 mg USD 4000 Ask For Quote & Lead Time

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Description

Emraclidine is a muscarinic M4 receptor positive allosteric modulator (WO2018002760, compound 11). Emraclidine can be used for the research of neurological diseases[1].

IC50 & Target

Muscarinic M4 Receptor[1]

In Vitro

Emraclidine is a muscarinic M4 receptor positive allosteric modulator[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

390.40

Formula

C₂₀H₂₁F₃N₄O

CAS No.
Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Solvent & Solubility
In Vitro: 

DMSO : 25 mg/mL (64.04 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.5615 mL 12.8074 mL 25.6148 mL
5 mM 0.5123 mL 2.5615 mL 5.1230 mL
10 mM 0.2561 mL 1.2807 mL 2.5615 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.5 mg/mL (6.40 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.5 mg/mL (6.40 mM); Clear solution

*All of the co-solvents are provided by MCE.
References
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  • Molarity Calculator

  • Dilution Calculator

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This equation is commonly abbreviated as: C1V1 = C2V2

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× = ×
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Product Name:
Emraclidine
Cat. No.:
HY-132812
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