ENPP3 Inhibitor 1
Based on 1 Customer Validation
ENPP3 Inhibitor 1 is a selective inhibitor of ENPP3, with IC50s of 0.15 µM (ENPP3) and 41.4 µM (ENPP1) respectively. ENPP3 Inhibitor 1 shows anti-tumor activities against breast cancer and cervical cancer.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- Reinheit: 99.43%
- CAS. Nr.: 2803505-90-8
- Formel: C20H14F3NO5S
- Molecular Weight:437.39
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Speicherung:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
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Biologische Aktivität
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Chemical Information
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Lösungsmittel & Löslichkeit
- Reinheit & Dokumentation
- Verweise
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Help & FAQs
Biologische Aktivität
Beschreibung
In Vitro
ENPP3 Inhibitor 1 (Compound 4t) (100 μM, 24 h) shows anti-tumor activities against human cancer cell lines MCF7, HeLa and human embryonic kidney cell lines HEK293, with the inhibition rate of 29.6%, 49.7% and 8.6%[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS. Nr. 2803505-90-8
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Appearance Solid
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Molecular Weight 437.39
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Formel C20H14F3NO5S
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Color White to off-white
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SMILES
O=C(C1=CC=CC=C1)NC2=CC=C(C=C2)OS(=O)(C3=CC=C(C=C3)OC(F)(F)F)=O
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Lösungsmittel & Löslichkeit
In Vitro:
DMSO : ≥ 116.67 mg/mL (266.74 mM; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
* "≥" means soluble, but saturation unknown.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
Reinheit & Dokumentation
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Data Sheet (270 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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Handling Instructions (2659 KB)
Verweise
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.2863 mL | 11.4314 mL | 22.8629 mL | 57.1572 mL |
| 5 mM | 0.4573 mL | 2.2863 mL | 4.5726 mL | 11.4314 mL | |
| 10 mM | 0.2286 mL | 1.1431 mL | 2.2863 mL | 5.7157 mL | |
| 15 mM | 0.1524 mL | 0.7621 mL | 1.5242 mL | 3.8105 mL | |
| 20 mM | 0.1143 mL | 0.5716 mL | 1.1431 mL | 2.8579 mL | |
| 25 mM | 0.0915 mL | 0.4573 mL | 0.9145 mL | 2.2863 mL | |
| 30 mM | 0.0762 mL | 0.3810 mL | 0.7621 mL | 1.9052 mL | |
| 40 mM | 0.0572 mL | 0.2858 mL | 0.5716 mL | 1.4289 mL | |
| 50 mM | 0.0457 mL | 0.2286 mL | 0.4573 mL | 1.1431 mL | |
| 60 mM | 0.0381 mL | 0.1905 mL | 0.3810 mL | 0.9526 mL | |
| 80 mM | 0.0286 mL | 0.1429 mL | 0.2858 mL | 0.7145 mL | |
| 100 mM | 0.0229 mL | 0.1143 mL | 0.2286 mL | 0.5716 mL |
ENPP3 Inhibitor 1 Related Classifications
HY-169804 Related Classifications
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