KSK68
KSK68 is a high-affinity dual sigma-1 and histamine H3 receptor antagonist, with Kis of 7.7, 3.6, 22.4 nM for H3 receptor, sigma-1, sigma-2 receptor respectively. KSK68 has negligible affinity at the other histamine receptor subtypes. KSK68 can be used for research of nociceptive and neuropathic pain.
For research use only. We do not sell to patients.
- CAS No.: 2566715-91-9
- Formula: C23H28N2O2
- Molecular Weight:364.48
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
7.7 nM, 3.6 nM、22.4 nM (H3 receptor, sigma-1, sigma-2 receptor)[1]
Chemical Information
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CAS No. 2566715-91-9
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Molecular Weight 364.48
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Formula C23H28N2O2
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SMILES
O=C(C1CC1)C2=CC=C(OCCCN3CCC(C4=CC=NC=C4)CC3)C=C2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)