LAS38096
LAS38096 is a potent, selective, and efficacious A2B Adenosine Receptor antagonist, with a Ki of 17 nM.
For research use only. We do not sell to patients.
- CAS No.: 851371-22-7
- Formula: C17H12N6O
- Molecular Weight:316.32
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All Adenosine Receptor Isoforms
More
Biological Activity
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A2B 17 nM (Ki) |
A1 >1000 nM (Ki) |
A2A >2500 nM (Ki) |
A3 >1000 nM (Ki) |
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| CHO | IC50 |
349 nM
Compound: 5, LAS38096
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Activity at mouse A2B receptor expressed in CHO cells assessed as inhibition of NECA-induced intracellular cAMP levels by ELISA
Activity at mouse A2B receptor expressed in CHO cells assessed as inhibition of NECA-induced intracellular cAMP levels by ELISA
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[PMID: 17469811] |
| HEK293 | IC50 |
321 nM
Compound: 5, LAS38096
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Activity at human A2B receptor expressed in HEK293 cells assessed as inhibition of NECA-induced intracellular cAMP levels by ELISA
Activity at human A2B receptor expressed in HEK293 cells assessed as inhibition of NECA-induced intracellular cAMP levels by ELISA
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[PMID: 17469811] |
Chemical Information
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CAS No. 851371-22-7
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Molecular Weight 316.32
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Formula C17H12N6O
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SMILES
C1(C2=CN=C(NC3=CC=CN=C3)N=C2C4=CC=CO4)=NC=NC=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
LAS38096 Related Classifications
HY-111295 Related Classifications
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