EN10
EN10 is a ligand for the muscle-specific E3 ligase KLHL41, which can be used to synthesize PROTAC KBD-1 (HY-184151) targeting BRD4.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 2093466-80-7
- Fòrmula: C21H23N3O
- Peso molecular:333.43
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Actividad biológica
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KLHL41 |
EN10 (5-15 μM; 30 min) selectively binds to KLHL41 (but not KLHL40) in live RH30 human muscle rhabdomyosarcoma cells[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 2093466-80-7
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Peso molecular 333.43
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Fòrmula C21H23N3O
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SMILES
[C@@H]1(C2=CC=CC=C2)OCC[C@H]1CNCC3=CNN=C3C4=CC=CC=C4
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)