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Referencia número: HY-14845

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Levomequitazine

(Synonyms: (S)-Mequitazine)

Levomequitazine (Compound V0114) ((S)-Mequitazine), the levorotatory enantiomer of Mequitazine (HY-B2168), is an orally active, inverse H4 receptor agonist (IC₅₀s: 94 nM (hM2), 17 nM (hM3)). Levomequitazine strongly binds to human histamine H4 receptor. Levomequitazine antagonizes the activating action induced by histamine on H4 receptor. Levomequitazine induces a powerful and statistically significant anti-inflammatory effect. Levomequitazine can be used for research on inflammatory diseases.

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No. CAS: 88598-74-7
Fòrmula: C₂₀H₂₂N₂S
Peso molecular:322.47

Almacenamiento:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (274 KB)

Levomequitazine Chemical Structure

No. CAS: 88598-74-7

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Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

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Descripciòn

IC₅₀ & Target

IC₅₀: 94 nM (hM2), 17 nM (hM3)^[1]

Ver todos los productos específicos de isoformas Histamine Receptor :

Chemical Information

No. CAS 88598-74-7
Peso molecular 322.47
Fòrmula C₂₀H₂₂N₂S
SMILES

N1(C2=CC=CC=C2SC3=CC=CC=C31)C[C@H]4C5CCN(CC5)C4
Synonyms

(S)-Mequitazine
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureza y Documentación

Select Batch:

Pureza: 99.98%

Assay: 99.98%

ee.: 99.98%

Ficha de datos (274 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instrucciones de manejo (2659 KB)

Referencias

[1]. Thierry Clerc, et al. Mequitazine for treating or preventing pathologies involving histamine h4 receptors. WO2009071625A1. WIPO (PCT). 2008-12-04.

Calculators

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How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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Levomequitazine

Ver todos los productos específicos de isoformas Histamine Receptor

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Chemical Information

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Referencias

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Levomequitazine Related Classifications

HY-14845 Related Classifications