MCL-524
MCL-524 is a highly selective full agonist of the dopamine D2 receptor with a Kd value of 1.34 nM. MCL-524 specifically binds to the high-affinity state of the dopamine D2 receptor; this binding is abolished by guanylylimidodiphosphate, and it can distinguish between D2high and D2low sites. MCL-524 is applicable to research related to Parkinson's disease and schizophrenia.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 1863967-01-4
- Fòrmula: C21H24FNO3
- Peso molecular:357.42
-
Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Actividad biológica
-
Chemical Information
- Pureza y Documentación
- Referencias
-
Help & FAQs
Ver todos los productos específicos de isoformas Dopamine Receptor
More
Actividad biológica
|
D2 Receptor 1.34 nM (Kd) |
MCL-524 competes with [3H]MCL-524 for binding to the human long-form D2 receptor expressed in CHO cells, with an inhibition constant (Ki) of 2.28 nM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
-
No. CAS 1863967-01-4
-
Peso molecular 357.42
-
Fòrmula C21H24FNO3
-
SMILES
OC1=CC=C2C(C3=C4C(CCN(CCC)[C@]4([H])C2)=CC(OCCF)=C3)=C1O
-
Envío
Room temperature in continental US; may vary elsewhere.
-
Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
MCL-524 Related Classifications
HY-184208 Related Classifications
Powered by Bioz