SR2595
SR2595 is an inverse agonist of PPARγ with an IC50 of 30 nM.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 1415252-61-7
- Fòrmula: C37H38N2O3
- Peso molecular:558.71
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Almacenamiento:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
Actividad biológica
Descripciòn
IC50 & Target
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PPARγ 30 nM (IC50) |
Cellular Effect
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Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| HEK-293T | EC50 |
355 nM
Compound: 51
|
Transactivation of human PPARgamma in HEK293T cells after 18 hrs by luciferase reporter gene assay
Transactivation of human PPARgamma in HEK293T cells after 18 hrs by luciferase reporter gene assay
|
[PMID: 26396687] |
Chemical Information
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No. CAS 1415252-61-7
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Appearance Solid
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Peso molecular 558.71
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Fòrmula C37H38N2O3
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Color Off-white to pink
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SMILES
CC(N1CC2=CC=C(C=C2)C3=CC=CC=C3C(O)=O)=C(C4=C1C=CC(C(N[C@H](C5=CC=C(C=C5)C(C)(C)C)C)=O)=C4)C
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)