GSK9311 hydrochloride
Based on 1 publication(s) in Google Scholar
GSK9311 hydrochloride, a less active analogue of GSK6853, can be used as a negative control. GSK9311 hydrochloride inhibits BRPF bromodomain with pIC50 values of 6.0 and 4.3 for BRPF1 and BRPF2, respectively.
For research use only. We do not sell to patients.
- CAS No.: 2253733-09-2
- Formula: C24H32ClN5O3
- Molecular Weight:474.00
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Publications Citing Use of MedChemExpress (MCE) GSK9311 hydrochloride
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Biological Activity
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BRPF1 6.0 (pIC50) |
BRPF2 4.3 (pIC50) |
GSK6853 is a potent (300 pM), soluble, cell active (20 nM), and highly selective inhibitor of the BRPF1 bromodomain, and demonstrates properties suitable for cellular and in vivo studies. GSK6853 is a less active analogue of GSK6853 in which the 5-amide is alkylated[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2253733-09-2
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Molecular Weight 474.00
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Formula C24H32ClN5O3
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SMILES
[H]Cl.C[C@@H]1CNCCN1C2=C(N(CC)C(C3=CC=CC=C3OC)=O)C=C(C(N4C)=C2)N(C)C4=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Publications (1)
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Journal Impact Factor
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Most Recent
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
GSK9311 hydrochloride Related Classifications
HY-100729A Related Classifications
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