Iferanserin hydrochloride
Iferanserin hydrochloride (S-MPEC hydrochloride) is a selective serotonin receptor antagonist with the potential to inhibit internal hemorrhoids. Iferanserin hydrochloride demonstrated efficacy and tolerability in ongoing Phase IIb clinical trials, with the ability to significantly reduce patient-reported symptoms of bleeding and pruritus.
For research use only. We do not sell to patients.
- CAS No.: 210350-29-1
- Formula: C23H29ClN2O
- Molecular Weight:384.94
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All 5-HT Receptor Isoforms
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Biological Activity
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5-HT2A Receptor |
Chemical Information
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CAS No. 210350-29-1
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Molecular Weight 384.94
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Formula C23H29ClN2O
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SMILES
CN(CCCC1)[C@@H]1CCC2=C(C=CC=C2)NC(/C=C/C3=CC=CC=C3)=O.Cl
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Synonyms
S-MPEC hydrochloride
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
[1]. Herold A, et al. Intra-anal Iferanserin 10 mg BID for hemorrhoid disease: a prospective, randomized, double-blind, placebo-controlled trial. Clin Ther. 2012 Feb;34(2):329-40. [Content Brief]
[2]. Intra-anal Iferanserin 10 mg BID for hemorrhoid disease: a prospective, randomized, double-blind, placebo-controlled trial [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)