U-99363E
U-99363E is a selective dopamine D4 receptor antagonist with a Ki value of 2.2 nM. U-99363E exhibits at least 100-fold lower affinity for other dopaminergic, serotonergic and adrenergic receptors. U-99363E can be used in studies related to selective dopamine D4 site labeling or blockade.
For research use only. We do not sell to patients.
- CAS No.: 170856-57-2
- Formula: C20H27N3O
- Molecular Weight:325.45
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Description
IC50 & Target
[1]|
Human D4 Receptor 2.2 nM (Ki) |
In Vitro
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 170856-57-2
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Molecular Weight 325.45
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Formula C20H27N3O
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SMILES
CCOC1=CC=CN=C1N(C2CCN(CC2)CC3=CC=CC=C3)C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
U-99363E Related Classifications
HY-169136 Related Classifications
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Keywords
- U-99363E
- 170856-57-2
- Dopamine Receptor
- 17β-HSD
- 17beta-HSD
- 17β-hydroxysteroid dehydrogenases
- 17 beta-hydroxysteroid dehydrogenase
- Chinese hamster ovary cells
- human dopamine D4 receptor
- adrenergic receptors
- human embryonic kidney cell membranes
- rat D2? dopamine receptors
- mammalian cells
- serotonergic receptors
- dopaminergic receptors
- quinpirole
- Inhibitor
- inhibitor
- inhibit