PGN-9856
Based on 1 Customer Validation
PGN-9856 is a selective and high affinity (pKi ≥ 8.3) ligand at EP2 receptor. PGN-9856 is a potetn and non-prostanoid EP2 receptor agonist (pEC50 ≥ 8.5). PGN-9856 shows anti-inflammatory and anti-glaucoma activities.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度 : 98.90%
- CAS 番号: 863704-91-0
- 分子式: C21H15F2NO4
- 分子量:383.34
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保管条件:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
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溶剤 & 溶解度
- プロトコル
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
生物活性
製品説明
IC50 & Target
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EP2 ≥ 8.5 (pEC50) |
EP2 ≥ 8.3 (pKi) |
化学情報
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CAS 番号 863704-91-0
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性状 Solid
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分子量 383.34
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分子式 C21H15F2NO4
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Color White to off-white
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SMILES
O=C(O)COC1=CC=CC(NC(C2=CC(C3=CC=CC(F)=C3)=CC=C2F)=O)=C1
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
溶剤 & 溶解度
体外:
DMSO : 125 mg/mL (326.08 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
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データシート (268 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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取扱説明書 (2659 KB)
参考文献
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.6087 mL | 13.0433 mL | 26.0865 mL | 65.2163 mL |
| 5 mM | 0.5217 mL | 2.6087 mL | 5.2173 mL | 13.0433 mL | |
| 10 mM | 0.2609 mL | 1.3043 mL | 2.6087 mL | 6.5216 mL | |
| 15 mM | 0.1739 mL | 0.8696 mL | 1.7391 mL | 4.3478 mL | |
| 20 mM | 0.1304 mL | 0.6522 mL | 1.3043 mL | 3.2608 mL | |
| 25 mM | 0.1043 mL | 0.5217 mL | 1.0435 mL | 2.6087 mL | |
| 30 mM | 0.0870 mL | 0.4348 mL | 0.8696 mL | 2.1739 mL | |
| 40 mM | 0.0652 mL | 0.3261 mL | 0.6522 mL | 1.6304 mL | |
| 50 mM | 0.0522 mL | 0.2609 mL | 0.5217 mL | 1.3043 mL | |
| 60 mM | 0.0435 mL | 0.2174 mL | 0.4348 mL | 1.0869 mL | |
| 80 mM | 0.0326 mL | 0.1630 mL | 0.3261 mL | 0.8152 mL | |
| 100 mM | 0.0261 mL | 0.1304 mL | 0.2609 mL | 0.6522 mL |
PGN-9856 関連分類
HY-115462 関連分類
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