country

Change Language

EN - English
FR - Français
DE - Deutsch
ES - Español
JA - 日本語
KO - 한국어

Product Name	Size / Unit Price	Qty

Total: USD 0.00 Checkout

Cat. No.: HY-182714

Copy Link Print Information

N 0840

(Synonyms: N6-Cyclopentyl-9-methyladenine)

N 0840 is a neutral antagonist of adenosine A₁ receptor (A₁AR), with a K_i value of 279 nM in rats and 1185 nM in humans. N 0840 modulates adenosine A₁ receptor to increase forskolin-induced cyclic 3′,5′-adenosine monophosphate production, with a GTP shift value close to 1. N 0840 can be used in studies of neuroprotection, cardiovascular/renal function^[1].

연구목적의 판매만을 진행합니다. 환자를 대상으로 한 판매는 하지 않습니다.

CAS No.: 109292-91-3
화학식: C₁₁H₁₅N₅
분자량:217.27

보관:

Please store the product under the recommended conditions in the Certificate of Analysis.

N 0840 Chemical Structure

CAS No.: 109292-91-3

사이즈

가격

재고

수량

Amount: USD 0.00

* 장바구니에 담기 전 물품의 수량을 선택해 주십시오.

Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- 제품 설명
- In Vitro
Chemical Information
순도&문서
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

제품 설명

All Adenosine Receptor Isoforms :

In Vitro

N 0840 binds to rat cortical membrane adenosine A₁ receptors with a K_i of 279 nM, and exhibits a GTP shift of 0.94^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 109292-91-3
분자량 217.27
화학식 C₁₁H₁₅N₅
SMILES

CN1C=NC2=C1N=CN=C2NC3CCCC3
Synonyms

N6-Cyclopentyl-9-methyladenine
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.

순도&문서

Handling Instructions (2659 KB)

References

[1]. Van Calenbergh S, et al. 5 ‘-Deoxy Congeners of 9-(3-Amido-3-deoxy-β-d-xylofuranosyl)-N 6-cyclopentyladenine: New Adenosine A1 Receptor Antagonists and Inverse Agonists. Journal of medicinal chemistry. 2002 Apr 25;45(9):1845-52.

Calculators

몰농도 계산기

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

농도 희석 계산기

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

MOQ

Minimum order quantity

100 mg

견적 받기 해외재고보유

Other size

견적 받기

Amount: USD 0.00

Biological Activity
- 제품 설명
- In Vitro
Chemical Information
순도&문서
References

상품명:
Cat. No.:
수량:
MCE Japan Authorized Agent:

상품명:
CAS No.:
Species:
Purity:
수량:

N 0840

All Adenosine Receptor Isoforms

Biological Activity

Chemical Information

순도&문서

References

Calculators

Help & FAQs

N 0840 Related Classifications

HY-182714 Related Classifications