SR2595
SR2595 is an inverse agonist of PPARγ with an IC50 of 30 nM.
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- CAS No.: 1415252-61-7
- 화학식: C37H38N2O3
- 분자량:558.71
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보관:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Protocol
- 순도&문서
- References
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Help & FAQs
Biological Activity
제품 설명
IC50 & Target
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PPARγ 30 nM (IC50) |
Cellular Effect
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| HEK-293T | EC50 |
355 nM
Compound: 51
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Transactivation of human PPARgamma in HEK293T cells after 18 hrs by luciferase reporter gene assay
Transactivation of human PPARgamma in HEK293T cells after 18 hrs by luciferase reporter gene assay
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[PMID: 26396687] |
Chemical Information
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CAS No. 1415252-61-7
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분자량 558.71
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화학식 C37H38N2O3
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SMILES
CC(N1CC2=CC=C(C=C2)C3=CC=CC=C3C(O)=O)=C(C4=C1C=CC(C(N[C@H](C5=CC=C(C=C5)C(C)(C)C)C)=O)=C4)C
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Please store the product under the recommended conditions in the Certificate of Analysis.
Protocol
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Cell Cytotoxicity Assay
Cytotoxicity assays are usually based on the assessment of cell membrane damage, which can also be indirectly detected by measuring cell viability. Detection methods include MTT assay, CKK-8 assay, LDH assay and ATP assay, etc.
순도&문서
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
SR2595 Related Classifications
HY-116521 Related Classifications
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