2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor
  4. PF-03246799 monohydrochloride

PF-03246799 monohydrochloride is a potent and selective 5-HT2C receptor agonist with an EC50 of 190 nM and a Ki of 160 nM. PF-03246799 monohydrochloride shows selectivity for 5-HT2C over 5-HT2A and 5-HT2B receptors. PF-03246799 monohydrochloride has the potential for stress urinary incontinence (SUI) research.

For research use only. We do not sell to patients.

PF-03246799 monohydrochloride

PF-03246799 monohydrochloride Chemical Structure

CAS No. : 1613666-08-2

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Other Forms of PF-03246799 monohydrochloride:

PF-03246799 monohydrochloride Related Antibodies

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Description

PF-03246799 monohydrochloride is a potent and selective 5-HT2C receptor agonist with an EC50 of 190 nM and a Ki of 160 nM. PF-03246799 monohydrochloride shows selectivity for 5-HT2C over 5-HT2A and 5-HT2B receptors. PF-03246799 monohydrochloride has the potential for stress urinary incontinence (SUI) research[1].

IC50 & Target[1]

5-HT2C Receptor

190 nM (EC50)

5-HT2C Receptor

160 nM (Ki)

Molecular Weight

275.78

Formula

C15H18ClN3
CAS No.
SMILES

C12=NC(CC3=CC=CC=C3)=NC=C1CCNCC2.Cl
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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PF-03246799 monohydrochloride Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PF-03246799 monohydrochloride1613666-08-25-HT ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorInhibitorinhibitorinhibit

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PF-03246799 monohydrochloride
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