1. GPCR/G Protein
    Neuronal Signaling
  2. Dopamine Receptor
  3. SB-277011

SB-277011 (Synonyms: SB-277011A)

Cat. No.: HY-10847
Handling Instructions

SB-277011 is a potent and delective dopamine D3 receptor antagonist (pKi values are 8.0, 6.0, 5.0 and <5.2 for D3, D2, 5-HT1D and 5-HT1B respectively); brain penetrant.

For research use only. We do not sell to patients.

SB-277011 Chemical Structure

SB-277011 Chemical Structure

CAS No. : 215803-78-4

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Description

SB-277011 is a potent and delective dopamine D3 receptor antagonist (pKi values are 8.0, 6.0, 5.0 and <5.2 for D3, D2, 5-HT1D and 5-HT1B respectively); brain penetrant. IC50 value: 8.0 (pKi) Target: D3 receptor

Molecular Weight

438.56

Formula

C₂₈H₃₀N₄O

CAS No.

215803-78-4

SMILES

O=C(C1=CC=NC2=CC=CC=C21)N[[email protected]@H]3CC[[email protected]](CC3)CCN4CC5=C(CC4)C=C(C#N)C=C5

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

SB-277011SB-277011ASB277011SB 277011Dopamine ReceptorInhibitorinhibitorinhibit

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