Sergolexole maleate
Sergolexole maleate is a potent 5-HT2 receptor antagonist. Sergolexole maleate antagonizes serotonin-amplified platelet aggregation.
For research use only. We do not sell to patients.
- CAS No.: 108674-87-9
- Formula: C30H40N2O7
- Molecular Weight:540.65
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All 5-HT Receptor Isoforms
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Biological Activity
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5-HT2 Receptor |
Chemical Information
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CAS No. 108674-87-9
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Molecular Weight 540.65
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Formula C30H40N2O7
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SMILES
OC(/C=C\C(O)=O)=O.CC(N1C2=C3C([C@]4([H])[C@@](N(C[C@@H](C4)C(O[C@@H]5CC[C@H](CC5)OC)=O)C)([H])CC3=C1)=CC=C2)C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
[1]. Cohen ML, et al. 5-Hydroxytryptamine2 receptor antagonist activity of the acid metabolite (1-isopropyl dihydrolysergic acid) of the ergoline ester, sergolexole (LY281067). J Pharmacol Exp Ther. 1989 Dec;251(3):1006-11. [Content Brief]
[2]. McBride PA, et al. Inhibition of serotonin-amplified human platelet aggregation by ketanserin, ritanserin, and the ergoline 5HT2 receptor antagonists-LY53857, sergolexole, and LY237733. Life Sci. 1990;47(23):2089-95. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Sergolexole maleate Related Classifications
HY-106324A Related Classifications
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