Tankyrase-IN-3
Tankyrase-IN-3 is a tankyrase 1 (TNKS1) inhibitor with an IC50 value of 22 nM. Tankyrase-IN-3 can be used for the research of cancer.
For research use only. We do not sell to patients.
- CAS No.: 938893-79-9
- Formula: C21H21N5O4
- Molecular Weight:407.42
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Description
IC50 & Target
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TNKS1 22 nM (IC50) |
In Vitro
Tankyrase-IN-3 has TNKS1 inhibition activity with an IC50 value of 22 nM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. Further protocols information, click here.
Chemical Information
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CAS No. 938893-79-9
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Molecular Weight 407.42
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Formula C21H21N5O4
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SMILES
O=C(OCC(N1CCN(CC1)C2=CC=CC=N2)=O)CC(C3=CC=CC=C34)=NNC4=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Protocols
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Cell Cytotoxicity Assay
Cytotoxicity assays are usually based on the assessment of cell membrane damage, which can also be indirectly detected by measuring cell viability. Detection methods include MTT assay, CKK-8 assay, LDH assay and ATP assay, etc.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)