1. GPCR/G Protein
  2. LPL Receptor

ASP-4058 

Cat. No.: HY-111021
Handling Instructions

ASP-4058 is a next-generation, selective and oral bioactive agonist for Sphingosine 1-Phosphate receptors 1 and 5 (S1P1 and S1P5), ameliorates rodent experimental autoimmune encephalomyelitis with a favorable safety profile.

For research use only. We do not sell to patients.

ASP-4058 Chemical Structure

ASP-4058 Chemical Structure

CAS No. : 952565-91-2

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  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

ASP-4058 is a next-generation, selective and oral bioactive agonist for Sphingosine 1-Phosphate receptors 1 and 5 (S1P1 and S1P5), ameliorates rodent experimental autoimmune encephalomyelitis with a favorable safety profile[1].

IC50 & Target

S1P1 and S1P5[1].

Solvent & Solubility
In Vitro: 

10 mM in DMSO

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.2609 mL 11.3043 mL 22.6086 mL
5 mM 0.4522 mL 2.2609 mL 4.5217 mL
10 mM 0.2261 mL 1.1304 mL 2.2609 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

442.31

Formula

C₁₉H₁₂F₆N₄O₂

CAS No.

952565-91-2

SMILES

C[[email protected]](OC1=CC=C(C2=NC(C3=CC=C4N=CNC4=C3)=NO2)C=C1C(F)(F)F)C(F)(F)F

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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Product Name:
ASP-4058
Cat. No.:
HY-111021
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ASP-4058

Cat. No.: HY-111021