2. GPCR/G Protein Neuronal Signaling Immunology/Inflammation
  3. Histamine Receptor
  4. Azacyclonol

Azacyclonol  (Synonyms: γ-pipradol)

Cat. No.: HY-B0530 Purity: 99.99%
COA Handling Instructions

Azacyclonol (γ-pipradol), a metabolite of Terfenadine, is a central depressant agent. Azacyclonol is a ganglion-blocking agent. Azacyclonol can be used to diminish psychoses-induced hallucinations.

For research use only. We do not sell to patients.

Azacyclonol Chemical Structure

Azacyclonol Chemical Structure

CAS No. : 115-46-8

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Solution
10 mM * 1 mL in DMSO USD 55 In-stock
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1 g USD 60 In-stock
5 g USD 84 In-stock
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Customer Review

Based on 1 publication(s) in Google Scholar

Azacyclonol Related Antibodies

Top Publications Citing Use of Products

1 Publications Citing Use of MCE Azacyclonol

  • Biological Activity

  • Purity & Documentation

  • References

  • Customer Review

Description

Azacyclonol (γ-pipradol), a metabolite of Terfenadine, is a central depressant agent. Azacyclonol is a ganglion-blocking agent. Azacyclonol can be used to diminish psychoses-induced hallucinations[1][2][3].

In Vitro

Azacyclonol is formed from Terfenadine in rat liver[2].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Azacyclonol Related Antibodies
In Vivo

Azacyclonol causes depressed activity in mice and rats[3].
Azacyclonol antagonizes increased coordination activity in mice induced by pipradrol, amphetamine, morphine and cocaine and prolongs Hexobarbital hypnosis[3].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.
Molecular Weight

267.37

Appearance

Solid

Formula

C18H21NO
CAS No.
SMILES

OC(C1=CC=CC=C1)(C2CCNCC2)C3=CC=CC=C3
Shipping

Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (374.01 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 3.7401 mL 18.7007 mL 37.4014 mL
5 mM 0.7480 mL 3.7401 mL 7.4803 mL
10 mM 0.3740 mL 1.8701 mL 3.7401 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.5 mg/mL (9.35 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.5 mg/mL (9.35 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.5 mg/mL (9.35 mM); Clear solution

*All of the co-solvents are available by MCE.
Purity & Documentation
References
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Azacyclonol Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

Azacyclonol115-46-8γ-pipradolHistamine ReceptorTerfenadinecentraldepressantpsychoseshallucinationsInhibitorinhibitorinhibit

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