1. Membrane Transporter/Ion Channel
    Neuronal Signaling
  2. Calcium Channel
  3. Bepridil hydrochloride

Bepridil hydrochloride (Synonyms: CERM 1978)

Cat. No.: HY-103315 Purity: 99.76%
Handling Instructions

Bepridil hydrochloride (CERM 1978) is a calcium channel blocker, with antianginal activity.

For research use only. We do not sell to patients.

Bepridil hydrochloride Chemical Structure

Bepridil hydrochloride Chemical Structure

CAS No. : 68099-86-5

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 55 In-stock
Estimated Time of Arrival: December 31
5 mg USD 50 In-stock
Estimated Time of Arrival: December 31
10 mg USD 70 In-stock
Estimated Time of Arrival: December 31
50 mg   Get quote  
100 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

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Description

Bepridil hydrochloride (CERM 1978) is a calcium channel blocker, with antianginal activity.

IC50 & Target

Calcium channel[1]

In Vitro

Bepridil hydrochloride is a calcium channel blocker, with antianginal activity[1].

In Vivo

Bepridil hydrochloride (21 mg/kg) reduces heart rate and mean arterial pressure, decreases the mean coronary vascular resistance and increases stroke volume in rats[1].

Molecular Weight

403.00

Formula

C₂₄H₃₅ClN₂O

CAS No.

68099-86-5

SMILES

[H]Cl.CC(C)COCC(N1CCCC1)CN(C2=CC=CC=C2)CC3=CC=CC=C3

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : ≥ 150 mg/mL (372.21 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.4814 mL 12.4069 mL 24.8139 mL
5 mM 0.4963 mL 2.4814 mL 4.9628 mL
10 mM 0.2481 mL 1.2407 mL 2.4814 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.5 mg/mL (6.20 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.5 mg/mL (6.20 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.5 mg/mL (6.20 mM); Clear solution

*All of the co-solvents are provided by MCE.
References

Purity: 99.76%

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  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

BepridilCERM 1978CERM1978CERM-1978Calcium ChannelCa2+ channelsCa channelsInhibitorinhibitorinhibit

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Product name:
Bepridil hydrochloride
Cat. No.:
HY-103315
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