1. Metabolic Enzyme/Protease
  2. RAR/RXR

Trifarotene (Synonyms: CD5789)

Cat. No.: HY-100256
Handling Instructions

Trifarotene is a retinoic acid receptor (RAR) agonist with Kdapp of 2, 15 and 500 nM for RARγ, RARβ and RARα, respectively.

For research use only. We do not sell to patients.

Trifarotene Chemical Structure

Trifarotene Chemical Structure

CAS No. : 895542-09-3

Size Price Stock
1 mg USD 1502 Get quote
5 mg USD 2404 Get quote
10 mg USD 3847 Get quote

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Customer Review

  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

Trifarotene is a retinoic acid receptor (RAR) agonist with Kdapp of 2, 15 and 500 nM for RARγ, RARβ and RARα, respectively.

IC50 & Target

Kdapp: 2 nM (RARγ), 15 nM (RARβ), 500 nM (RARα)[1]

Clinical Trial
Solvent & Solubility
In Vitro: 

10 mM in DMSO

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.1759 mL 10.8795 mL 21.7590 mL
5 mM 0.4352 mL 2.1759 mL 4.3518 mL
10 mM 0.2176 mL 1.0879 mL 2.1759 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

459.58

Formula

C₂₉H₃₃NO₄

CAS No.

895542-09-3

SMILES

O=C(C1=CC=C(C2=CC=C(OCCO)C(C3=CC=C(N4CCCC4)C(C(C)(C)C)=C3)=C2)C=C1)O

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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This equation is commonly abbreviated as: C1V1 = C2V2

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× = ×
C1   V1   C2   V2

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Product Name:
Trifarotene
Cat. No.:
HY-100256
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Trifarotene

Cat. No.: HY-100256