DCE_254
DCE_254 is an EZH2 inhibitor (IC50=11 μM) that also exhibits significant antiproliferative activity against lymphoma cell lines. DCE_254 inhibits the development of hypermethylation-related cancers by inhibiting the SAM-mediated methyl transfer process (IC50=10.3 μM).
For research use only. We do not sell to patients.
- CAS No.: 673443-80-6
- Formula: C21H17N9OS
- Molecular Weight:443.48
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Histone Methyltransferase Isoforms
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Biological Activity
Chemical Information
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CAS No. 673443-80-6
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Molecular Weight 443.48
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Formula C21H17N9OS
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SMILES
O=C1N=C(NC(CSC2=NN=NN2C3=CC=CC=C3)=C1)NC4=NC(C)=C5C=CC=CC5=N4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)