BRD4 Inhibitor-34
Based on 1 Customer Validation
BRD4 Inhibitor-34 (Compound 12a) is a BRD4 inhibitor with an IC50 of 24 μM.
For research use only. We do not sell to patients.
- Purity: 96.84%
- CAS No.: 1095051-68-5
- Formula: C9H6ClNOS
- Molecular Weight:211.67
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Storage:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
Biological Activity
IC50: 24 μM (BRD4)[1].
Chemical Information
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CAS No. 1095051-68-5
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Appearance Solid
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Molecular Weight 211.67
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Formula C9H6ClNOS
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Color Off-white to light brown
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SMILES
O=C1SC=C(C2=CC=CC(Cl)=C2)N1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
DMSO : ≥ 150 mg/mL (708.65 mM; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
* "≥" means soluble, but saturation unknown.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (269 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 4.7243 mL | 23.6217 mL | 47.2434 mL | 118.1084 mL |
| 5 mM | 0.9449 mL | 4.7243 mL | 9.4487 mL | 23.6217 mL | |
| 10 mM | 0.4724 mL | 2.3622 mL | 4.7243 mL | 11.8108 mL | |
| 15 mM | 0.3150 mL | 1.5748 mL | 3.1496 mL | 7.8739 mL | |
| 20 mM | 0.2362 mL | 1.1811 mL | 2.3622 mL | 5.9054 mL | |
| 25 mM | 0.1890 mL | 0.9449 mL | 1.8897 mL | 4.7243 mL | |
| 30 mM | 0.1575 mL | 0.7874 mL | 1.5748 mL | 3.9369 mL | |
| 40 mM | 0.1181 mL | 0.5905 mL | 1.1811 mL | 2.9527 mL | |
| 50 mM | 0.0945 mL | 0.4724 mL | 0.9449 mL | 2.3622 mL | |
| 60 mM | 0.0787 mL | 0.3937 mL | 0.7874 mL | 1.9685 mL | |
| 80 mM | 0.0591 mL | 0.2953 mL | 0.5905 mL | 1.4764 mL | |
| 100 mM | 0.0472 mL | 0.2362 mL | 0.4724 mL | 1.1811 mL |