country

Change Language

EN - English
FR - Français
DE - Deutsch
ES - Español
JA - 日本語
KO - 한국어

Product Name	Size / Unit Price	Qty

Total: USD 0.00 Checkout

Cat. No.: HY-167160

Copy Link Print Information

AZ12099548

AZ12099548 is a TRPV1 antagonist. AZ12099548 inhibits both Capsaicin (HY-10448)- and low pH-induced calcium mobilization.

Nos produits utilisent uniquement pour la recherche. Nous ne vendons pas aux patients.

CAS No.: 790689-76-8
Formule: C₁₉H₂₀N₂O₃S
Masse moléculaire:356.44

Stockage:

Please store the product under the recommended conditions in the Certificate of Analysis.

AZ12099548 Chemical Structure

CAS No.: 790689-76-8

Size

Prix

Stock

Quantité

Amount: USD 0.00

* Veuillez sélectionner la quantité avant d'ajouter des articles.

Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- IC₅₀ & Target
- In Vitro
Chemical Information
Pureté et documentation
Références
Calculators
Help & FAQs
Classifications
Bioz

Activité biologique

Description

AZ12099548 is a TRPV1 antagonist. AZ12099548 inhibits both Capsaicin (HY-10448)- and low pH-induced calcium mobilization^[1].

IC₅₀ & Target^[1]

hTRPV1

Voir tous les produits spécifiques à Isoform TRP Channel :

In Vitro

AZ12099548 (Compound AZ C) inhibits both Capsaicin (HY-10448)- and low pH-induced calcium mobilization in human TRPV1-expressing cells, with IC₅₀ values of 10 nM and 22 nM, respectively^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 790689-76-8
Masse moléculaire 356.44
Formule C₁₉H₂₀N₂O₃S
SMILES

O=C(NC=1C=CC=2SC(=NC2C1)CO)C3=CC=C(OC(C)(C)C)C=C3
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Instruction de manipulation (2659 KB)

Références

[1]. Cuypers E, et al. Transient receptor potential vanilloid 1 and xenobiotics. CNS Neurol Disord Drug Targets. 2008;7(2):159-171. [Content Brief]

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Calculateur de dilution

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

100 mg

Obtenir un devis En stock

Amount: USD 0.00

Activité biologique
- Description
- IC₅₀ & Target
- In Vitro
Chemical Information
Pureté et documentation
Références

Nom du produit:
Cat. No.:
Quantité:
MCE Japan Authorized Agent:

Nom du produit:
CAS No.:
Species:
Pureté:
Quantité:

AZ12099548

Voir tous les produits spécifiques à Isoform TRP Channel

Activité biologique

Chemical Information

Pureté et documentation

Références

Calculators

Help & FAQs

AZ12099548 Related Classifications

HY-167160 Related Classifications