N 0840
N 0840 is a neutral antagonist of adenosine A1 receptor (A1AR), with a Ki value of 279 nM in rats and 1185 nM in humans. N 0840 modulates adenosine A1 receptor to increase forskolin-induced cyclic 3′,5′-adenosine monophosphate production, with a GTP shift value close to 1. N 0840 can be used in studies of neuroprotection, cardiovascular/renal function[1].
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- CAS No.: 109292-91-3
- Formule: C11H15N5
- Masse moléculaire:217.27
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
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Activité biologique
N 0840 binds to rat cortical membrane adenosine A1 receptors with a Ki of 279 nM, and exhibits a GTP shift of 0.94[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 109292-91-3
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Masse moléculaire 217.27
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Formule C11H15N5
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SMILES
CN1C=NC2=C1N=CN=C2NC3CCCC3
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Synonyms
N6-Cyclopentyl-9-methyladenine
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
N 0840 Related Classifications
HY-182714 Related Classifications
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