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Cat. No.: HY-116882

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PIK-39

PIK-39 is a selective PI3Kδ inhibitor with an IC₅₀ of 0.30 μM. PIK-39 has a propeller-like structure that induces conformational changes in the ATP-binding region of its target. PIK-39 is applicable to the research of autoimmune diseases.

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CAS No.: 371242-53-4
Formule: C₂₁H₁₅ClN₆O₂S
Masse moléculaire:450.90

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Please store the product under the recommended conditions in the Certificate of Analysis.

PIK-39 Chemical Structure

CAS No.: 371242-53-4

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- IC₅₀ & Target
Chemical Information
Pureté et documentation
Références
Calculators
Help & FAQs
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Activité biologique

Description

IC₅₀ & Target^[1]

PI3Kδ

0.3 μM (IC₅₀)

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Chemical Information

CAS No. 371242-53-4
Masse moléculaire 450.90
Formule C₂₁H₁₅ClN₆O₂S
SMILES

O=C1N(C(CSC2=C3N=CNC3=NC=N2)=NC4=C1C(Cl)=CC=C4)C5=CC=CC=C5OC
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Instruction de manipulation (2659 KB)

Références

[1]. Cushing T D, et al. Discovery and in vivo evaluation of (S)-N-(1-(7-Fluoro-2-(pyridin-2-yl) quinolin-3-yl) ethyl)-9 H-purin-6-amine (AMG319) and related PI3Kδ inhibitors for inflammation and autoimmune disease[J]. Journal of Medicinal Chemistry, 2015, 58(1): 480-511.

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Calculateur de molarité

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Calculateur de dilution

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Activité biologique
- Description
- IC₅₀ & Target
Chemical Information
Pureté et documentation
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PIK-39

Voir tous les produits spécifiques à Isoform PI3K

Activité biologique

Chemical Information

Pureté et documentation

Références

Calculators

Help & FAQs

PIK-39 Related Classifications

HY-116882 Related Classifications