ST-CY14
ST-CY14 is an inhibitor for Nur77-PPARγ interaction with an EC50 of 3.15 μM, that binds to Nur77 (Kd=32 nM), blocks Nur77 from being ubiquitinated and degraded by PPARγ, reduces fatty acid uptake and mitochondrial respiration, and inhibits the transcription of CD36 and FABP4. ST-CY14 inhibits the proliferation and migration of cancer cell MCF7 and MDA-MB-231. ST-CY14 inhibits tumor growth and bone metastasis in mouse models.
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- Formule: C139H237N57O31S2
- Masse moléculaire:3266.86
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
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Activité biologique
Description
Chemical Information
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Masse moléculaire 3266.86
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Formule C139H237N57O31S2
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Sequence
Cys-Glu-Gly-Cys-Lys-Gly-Phe-{S5}-Arg-Arg-Thr-{S5}-Arg-Tyr-Tyr-Gly-Arg-Lys-Lys-Arg-Arg-Gln-Arg-Arg-Arg-NH2
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Sequence Shortening
CEGCKGF-{S5}-RRT-{S5}-RYYGRKKRRQRRR-NH2
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
ST-CY14 Related Classifications
HY-P10873 Related Classifications
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