Giclanfentrine
Giclanfentrine is a potent PDE3A inhibitor with an IC50 of 0.0058 μM. Giclanfentrine inhibits PDE4B1 activity with an IC50 of 12.9 μM. Giclanfentrine is applicable to studies related to PDE3/cAMP signaling.
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- CAS. Nr.: 2408152-69-0
- Formel: C30H35N7O5
- Molecular Weight:573.64
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
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Chemical Information
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Help & FAQs
Biologische Aktivität
Beschreibung
IC50 & Target
[1]|
PDE3A 0.0058 μM (IC50) |
PDE4B1 12.9 μM (IC50) |
In Vitro
Giclanfentrine (compound 23) inhibits the activities of recombinant PDE3A and PDE4B1 enzymes, with IC50 values of 0.0058 μM and 12.9 μM, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. .
Chemical Information
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CAS. Nr. 2408152-69-0
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Molecular Weight 573.64
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Formel C30H35N7O5
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SMILES
O=C(C1=C(N=NN1C)O)NCCN2/C(C=C3C4=C(CCN3C2=O)C=C(OCC)C(OC)=C4)=N/C5=C(C)C=C(C)C=C5C
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
Giclanfentrine Related Classifications
HY-171827 Related Classifications
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