PSB-1901
Based on 1 Customer Validation
PSB-1901 is a potent A2B adenosine receptor (A2BAR) antagonist with Kis of 0.0835 nM and 0.131 nM for human and mouse A2BARs respectively. PSB-1901 can be used for the research of cancer.
For research use only. We do not sell to patients.
- Purity: 96.33%
- CAS No.: 2332835-02-4
- Formula: C24H25BrN6O4S
- Molecular Weight:573.46
-
Storage:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
All Adenosine Receptor Isoforms
More
Biological Activity
Ki: 0.0835 nM (human A2BAR), 0.131 nM (mouse A2BAR)[1]
Chemical Information
-
CAS No. 2332835-02-4
-
Appearance Solid
-
Molecular Weight 573.46
-
Formula C24H25BrN6O4S
-
Color White to off-white
-
SMILES
O=C1NC2=C(C(N1CCC)=O)NC(C3=CC=C(S(=O)(N4CCN(CC4)C5=CC=C(C=C5)Br)=O)C=C3)=N2
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
DMSO : ≥ 100 mg/mL (174.38 mM; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
* "≥" means soluble, but saturation unknown.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
-
Data Sheet (268 KB)
-
SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
-
Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 1.7438 mL | 8.7190 mL | 17.4380 mL | 43.5950 mL |
| 5 mM | 0.3488 mL | 1.7438 mL | 3.4876 mL | 8.7190 mL | |
| 10 mM | 0.1744 mL | 0.8719 mL | 1.7438 mL | 4.3595 mL | |
| 15 mM | 0.1163 mL | 0.5813 mL | 1.1625 mL | 2.9063 mL | |
| 20 mM | 0.0872 mL | 0.4360 mL | 0.8719 mL | 2.1798 mL | |
| 25 mM | 0.0698 mL | 0.3488 mL | 0.6975 mL | 1.7438 mL | |
| 30 mM | 0.0581 mL | 0.2906 mL | 0.5813 mL | 1.4532 mL | |
| 40 mM | 0.0436 mL | 0.2180 mL | 0.4360 mL | 1.0899 mL | |
| 50 mM | 0.0349 mL | 0.1744 mL | 0.3488 mL | 0.8719 mL | |
| 60 mM | 0.0291 mL | 0.1453 mL | 0.2906 mL | 0.7266 mL | |
| 80 mM | 0.0218 mL | 0.1090 mL | 0.2180 mL | 0.5449 mL | |
| 100 mM | 0.0174 mL | 0.0872 mL | 0.1744 mL | 0.4360 mL |