1. Membrane Transporter/Ion Channel
  2. Sodium Channel
  3. DSP-2230

DSP-2230 

Cat. No.: HY-125079 Purity: 98.33%
Handling Instructions

DSP-2230 is a selective Nav1.7/Nav1.8 blocker.

For research use only. We do not sell to patients.

DSP-2230 Chemical Structure

DSP-2230 Chemical Structure

CAS No. : 1233231-30-5

Size Price Stock Quantity
Free Sample (0.5-1 mg)   Apply now  
10 mM * 1  mL in DMSO USD 111 In-stock
Estimated Time of Arrival: December 31
5 mg USD 120 In-stock
Estimated Time of Arrival: December 31
10 mg USD 200 In-stock
Estimated Time of Arrival: December 31
25 mg USD 400 In-stock
Estimated Time of Arrival: December 31
50 mg USD 650 In-stock
Estimated Time of Arrival: December 31
100 mg USD 1050 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

Based on 1 publication(s) in Google Scholar

Top Publications Citing Use of Products
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Description

DSP-2230 is a selective Nav1.7/Nav1.8 blocker[1][2].

IC50 & Target

Nav1.7/Nav1.8[1]

Molecular Weight

419.40

Formula

C₂₀H₂₀F₃N₅O₂

CAS No.

1233231-30-5

SMILES

C[[email protected]](NCC1=NC2=CC=C(OC3=CC(F)=C(F)C(F)=C3)N=C2N1C4CCC4)C(N)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 125 mg/mL (298.04 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.3844 mL 11.9218 mL 23.8436 mL
5 mM 0.4769 mL 2.3844 mL 4.7687 mL
10 mM 0.2384 mL 1.1922 mL 2.3844 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.25 mg/mL (5.36 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.25 mg/mL (5.36 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.25 mg/mL (5.36 mM); Clear solution

*All of the co-solvents are provided by MCE.
References

Purity: 98.33%

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  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

DSP-2230DSP2230DSP 2230Sodium ChannelNa channelsNa+ channelsInhibitorinhibitorinhibit

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Product name:
DSP-2230
Cat. No.:
HY-125079
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