DTP348
DTP348 is an inhibitor for carbonic anhydrase IX with a Ki of 8.3 nM in vitro and an IC50 of 19.26 μM in Xenopus oocytes. DTP348 exhibits slight toxicity in zebrafish embryos with LD50 of 3.5 mM. DTP348 can be used in the anti-cancer research.
For research use only. We do not sell to patients.
- CAS No.: 1383370-92-0
- Formula: C6H11N5O4S
- Molecular Weight:249.25
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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CA IX 8.3 nM (Ki) |
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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CAS No. 1383370-92-0
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Molecular Weight 249.25
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Formula C6H11N5O4S
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SMILES
O=S(NCCN1C([N+]([O-])=O)=CN=C1C)(N)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)