AH081
AH081 (Compound 38) is a CK1δ/ε PROTAC degrader. AH081 is the negative control compound of AH078 (HY-170859). AH081 has inhibitory but no degradation activity for CK1δ/ε by using an inactive stereoisomer of the VHL ligand. Pink: CK1δ/ε ligand (HY-148251); Blue: VHL ligase ligand (HY-125845B); Black: linker
(Pink: CK1δ and CK1ε ligand (HY-148251); Blue: VHL ligand (HY-125845B); Black: linker).
Para uso exclusivo en investigación. No vendemos a pacientes.
- Fòrmula: C51H60F2N10O5S
- Peso molecular:963.15
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
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Chemical Information
- Pureza y Documentación
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Help & FAQs
Ver todos los productos específicos de isoformas PROTACs
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Actividad biológica
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CK1δ |
CK1ε |
Chemical Information
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Peso molecular 963.15
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Fòrmula C51H60F2N10O5S
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SMILES
O=C(NCC1=CC=C(C=C1)C2=C(N=CS2)C)[C@H]3N(C[C@H](C3)O)C([C@H](C(C)(C)C)NC(CCCCCCC(N4CCC(F)(CC4)CN5C(C6=C7C(NC=C7)=NC=C6)=C(N=C5)C8=NC=C(C=C8)F)=O)=O)=O
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
AH081 Related Classifications
HY-170859A Related Classifications
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