N 0840
N 0840 is a neutral antagonist of adenosine A1 receptor (A1AR), with a Ki value of 279 nM in rats and 1185 nM in humans. N 0840 modulates adenosine A1 receptor to increase forskolin-induced cyclic 3′,5′-adenosine monophosphate production, with a GTP shift value close to 1. N 0840 can be used in studies of neuroprotection, cardiovascular/renal function[1].
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 109292-91-3
- Fòrmula: C11H15N5
- Peso molecular:217.27
-
Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Actividad biológica
-
Chemical Information
- Pureza y Documentación
- Referencias
-
Help & FAQs
Ver todos los productos específicos de isoformas Adenosine Receptor
More
Actividad biológica
N 0840 binds to rat cortical membrane adenosine A1 receptors with a Ki of 279 nM, and exhibits a GTP shift of 0.94[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
-
No. CAS 109292-91-3
-
Peso molecular 217.27
-
Fòrmula C11H15N5
-
SMILES
CN1C=NC2=C1N=CN=C2NC3CCCC3
-
Synonyms
N6-Cyclopentyl-9-methyladenine
-
Envío
Room temperature in continental US; may vary elsewhere.
-
Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
N 0840 Related Classifications
HY-182714 Related Classifications
Powered by Bioz