TOPORS - TOP1 binding arginine/serine rich protein, E3 ubiquitin ligase Gene
Species: Sus scrofa
Gene Type: protein coding
Gene ID: 100513812
TOPORS Products (3)
| mRNA | Protein | Name |
|---|---|---|
| XM_013980194.2 | XP_013835648.1 | E3 ubiquitin-protein ligase Topors isoform X2 |
| XM_005668076.3 | XP_005668133.1 | E3 ubiquitin-protein ligase Topors isoform X1 |
| XM_021064703.1 | XP_020920362.1 | E3 ubiquitin-protein ligase Topors isoform X3 |
| Protein Preferred Names | Protein Names | |
|---|---|---|
|
E3 ubiquitin-protein ligase Topors |
|
Related Agents
- Clinical Phase
- Pre-clinical Phase
Clinical Phase
Bioactive Molecules
(7)
| Cat. No. | Product Name |
Effect
|
Purity |
Phase |
|---|---|---|---|---|
| HY-164734 | Raludotatug Deruxtecan | 99.29% | Phase 3 | |
| HY-171689 | Puxitatug samrotecan | Inhibitor | 98.51% | Phase 2 |
| HY-168739 | Topoisomerase I inhibitor 17 | / | Phase 2 | |
| HY-171124 | Tilatamig samrotecan | Inhibitor | 95.26% | Phase 1 |
| HY-U00248 | LMP744 | Inhibitor | 98.33% | Phase 1 |
| HY-18350 | Indimitecan | Inhibitor | 98.30% | Phase 1 |
| HY-U00248A | LMP744 hydrochloride | Inhibitor | 99.08% | Phase 1 |
Pre-clinical Phase
Bioactive Molecules
(82)
| Cat. No. | Product Name |
Effect
|
Purity |
Rare Diseases
|
|---|---|---|---|---|
| HY-148819A | NH2-bicyclo[1.1.1]pentane-7-MAD-MDCPT hydrochloride | Inhibitor | 98.46% | Unkown |
| HY-148819 | NH2-bicyclo[1.1.1]pentane-7-MAD-MDCPT | Inhibitor | 98.71% | Unkown |
| HY-111630 | PluriSIn #2 | Inhibitor | 98.0% | Unkown |
| HY-118581 | Coralyne chloride | Inhibitor | 98.39% | Unkown |
| HY-174374 | Topobexin | Inhibitor | 99.04% | Unkown |
| HY-163099 | P5(PEG24)-VC-PAB-Exatecan | 99.74% | Unkown | |
| HY-153278 | Q901 | Inhibitor | 98.38% | Unkown |
| HY-164143 | T638 | Inhibitor | 98.61% | Unkown |
| HY-116785 | BRD32048 | Inhibitor | 99.94% | Unkown |
| HY-160005 | LMP517 | Inhibitor | 99.58% | Unkown |
| HY-153278A | Q901 TFA | Inhibitor | / | Unkown |
| HY-122594 | BNS-22 | Inhibitor | 99.50% | Unkown |
| HY-175203 | Topi MF-6 | Inhibitor | 99.79% | Unkown |
| HY-W008874 | meso-Tetra(4-pyridyl)porphine | Inhibitor | ≥97.0% | Unkown |
| HY-118911 | ATM Inhibitor-10 | Inhibitor | 98.7% | Unkown |
| HY-N0114A | (±)-Evodiamine | 99.74% | Unkown | |
| HY-123393 | PNU-142586 | Inhibitor | / | Unkown |
| HY-13550 | Ametantrone | Inhibitor | 97.28% | Unkown |
| HY-160857 | TOP5668 | Agonist | 98.07% | Unkown |
| HY-168489 | OBI-992 drug-linker | 96.64% | Unkown | |
| HY-RS14902 | TOPORS Human Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
| HY-RS14894 | TOP2A Human Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
| HY-126142 | Top1 inhibitor 1 | Inhibitor | 99.67% | Unkown |
| HY-RS14893 | TOP1MT Human Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
| HY-RS14897 | TOP2B Human Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
| HY-RS14899 | TOP3B Human Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
| HY-118942 | Topovale | Inhibitor | 99.94% | Unkown |
| HY-101115 | PI3K-IN-6 | Inhibitor | / | Unkown |
| HY-117142 | Quizalofop-P | Inhibitor | / | Unkown |
| HY-117613 | A-74932 hydrochloride | Inhibitor | / | Unkown |
| HY-120638 | BMS-250749 | Inhibitor | / | Unkown |
| HY-121560 | L-leucyldoxorubicin | / | Unkown | |
| HY-121866 | CP-84364 | Inhibitor | / | Unkown |
| HY-125387 | TOP1210 | / | Unkown | |
| HY-125426 | ToP-DNJ | Inhibitor | / | Unkown |
| HY-125500 | TOP1362 | Inhibitor | / | Unkown |
| HY-143265 | Topoisomerase I inhibitor 2 | / | Unkown | |
| HY-144222 | NSC 828467 | Inhibitor | / | Unkown |
| HY-144654 | HDAC/Top-IN-1 | Inhibitor | / | Unkown |
| HY-145851 | Top/HDAC-IN-1 | / | Unkown | |
| HY-145852 | Top/HDAC-IN-2 | / | Unkown | |
| HY-146437 | Topoisomerase I inhibitor 6 | Inhibitor | / | Unkown |
| HY-149348 | DiPT-4 | / | Unkown | |
| HY-159935 | Top1-IN-2 | Inhibitor | / | Unkown |
| HY-159966 | Top/HDAC-IN-3 | / | Unkown | |
| HY-160856 | TOP5300 | Agonist | / | Unkown |
| HY-161957 | Top1/2-IN-1 | Inhibitor | / | Unkown |
| HY-163118 | Topoisomerase II inhibitor 17 | / | Unkown | |
| HY-16560B | (R)-Camptothecin | Control | / | Unkown |
| HY-172259 | Toyaburgine | Inhibitor | / | Unkown |
| HY-173001 | AuL1 | Inhibitor | / | Unkown |
| HY-175700 | YCJ-02 | / | Unkown | |
| HY-175834 | DNA/TOP2A-IN-1 | / | Unkown | |
| HY-176762 | TOP3B-IN-1 | Inhibitor | / | Unkown |
| HY-178029 | RSK2/TOP2-IN-1 | / | Unkown | |
| HY-178036 | ZM484 | Inhibitor | / | Unkown |
| HY-180555 | SN38-(PEG)2-Pom-α | Activator | / | Unkown |
| HY-181080 | TOP1/TDP1-IN-1 | / | Unkown | |
| HY-18350A | Indimitecan hydrochloride | Inhibitor | / | Unkown |
| HY-184245 | Hsp90-IN-48 | Inhibitor | / | Unkown |
| HY-N15249 | 4"-Isovalerylspiramycin I | / | Unkown | |
| HY-N17442 | Echinoside A | / | Unkown | |
| HY-P11715 | Abz-GFDPFRQ-EDDnp | / | Unkown | |
| HY-P4926 | Mca-SEVKMDAEFRK(Dnp)RR-NH2 | / | Unkown | |
| HY-RS14890 | TOP1 Human Pre-designed siRNA Set A | / | Unkown | |
| HY-RS14891 | Top1 Mouse Pre-designed siRNA Set A | / | Unkown | |
| HY-RS14892 | Top1 Rat Pre-designed siRNA Set A | / | Unkown | |
| HY-RS14895 | Top2a Mouse Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
| HY-RS14896 | Top2a Rat Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
| HY-RS14898 | TOP3A Human Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
| HY-W654323 | PNU-142586 sodium | Inhibitor | / | Unkown |
| HY-W800535 | Cryptolepine | / | Unkown | |
| HY-133219 | Guajadial C | Inhibitor | / | Unkown |
| HY-160930 | TOP1288 | Inhibitor | / | Unkown |
| HY-169173 | AL284 | Inhibitor | / | Unkown |
| HY-180333 | Top-Tdp tri inhibitor C12 | / | Unkown | |
| HY-184297 | Topoisomerase II-IN-26 | Inhibitor | / | Unkown |
| HY-185300 | IKZF2-degrader 4 | Degrader | / | Unkown |
| HY-RS20119 | Top2b Mouse Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
| HY-RS21791 | Top3a Mouse Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
| HY-RS26623 | Top2b Rat Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
| HY-RS28307 | Top3a Rat Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
Bioactive MoleculesInhibitory Antibodies
(1)
| Cat. No. | Product Name |
Effect
|
Purity |
Rare Diseases
|
|---|---|---|---|---|
| HY-P990947 | Tilatamig | Inhibitor | 99.99% | Unkown |