KDR - kinase insert domain receptor Gene
Species: Macaca fascicularis
Gene Type: protein coding
Gene ID: 102136227
About KDR
Primary_assembly 5: 78,970,505-79,016,167 forward strand.Macaca_fascicularis_6.0:CM021943.1
This gene has 1 transcript (splice variant), 199 orthologues and 55 paralogues.
KDR Products (2)
| mRNA | Protein | Name |
|---|---|---|
| XM_005555270.3 | XP_005555327.2 | vascular endothelial growth factor receptor 2 |
| XM_005555270.3 | XP_005555327.2 | vascular endothelial growth factor receptor 2 |
| Protein Preferred Names | Protein Names | |
|---|---|---|
|
vascular endothelial growth factor receptor 2 |
|
Related Agents
- Approval
- Clinical Phase
- Pre-clinical Phase
Approval
Bioactive Molecules
(6)
| Cat. No. | Product Name |
Effect
|
Purity |
Rare Diseases
|
|---|---|---|---|---|
| HY-10260 | Vandetanib | 99.85% | Yes | |
| HY-112306 | Ripretinib | 98.90% | Yes | |
| HY-14914 | Azilsartan | 99.68% | Unkown | |
| HY-10330A | Toceranib phosphate | Inhibitor | 99.23% | Unkown |
| HY-10260B | Vandetanib hydrochloride | / | Unkown | |
| HY-10260A | Vandetanib trifluoroacetate | / | Unkown |
Clinical Phase
Bioactive Molecules
(14)
| Cat. No. | Product Name |
Effect
|
Purity |
Phase |
|---|---|---|---|---|
| HY-50751 | Linifanib | 99.39% | Phase 3 | |
| HY-10205 | Cediranib | 99.87% | Phase 3 | |
| HY-10203 | Vatalanib | Inhibitor | 99.93% | Phase 3 |
| HY-12018 | Vatalanib dihydrochloride | 99.68% | Phase 3 | |
| HY-13049 | Cediranib maleate | 99.95% | Phase 3 | |
| HY-12018A | Vatalanib hydrochloride | Inhibitor | / | Phase 3 |
| HY-110272 | Vatalanib succinate | Inhibitor | / | Phase 3 |
| HY-10374 | Semaxinib | Inhibitor | 99.92% | Phase 2 |
| HY-13024 | Rebastinib | 99.84% | Phase 2 | |
| HY-10338 | Foretinib | Inhibitor | 99.45% | Phase 2 |
| HY-10987A | ENMD-2076 | 99.99% | Phase 2 | |
| HY-10987 | ENMD-2076 Tartrate | 99.66% | Phase 2 | |
| HY-10204 | OSI-930 | 98.33% | Phase 1 | |
| HY-100315 | XL 999 | Inhibitor | 99.01% | Phase 1 |
Bioactive MoleculesInhibitory Antibodies
(2)
| Cat. No. | Product Name |
Effect
|
Purity |
Phase |
|---|---|---|---|---|
| HY-P99768 | Olinvacimab | Inhibitor | 95.00% | Phase 2 |
| HY-P991419 | MSB-0254 | Inhibitor | / | Phase 1 |
Pre-clinical Phase
Bioactive Molecules
(59)
| Cat. No. | Product Name |
Effect
|
Purity |
Rare Diseases
|
|---|---|---|---|---|
| HY-12299 | WH-4-023 | Inhibitor | 99.87% | Unkown |
| HY-151361 | AMPK-IN-3 | Inhibitor | 98.51% | Unkown |
| HY-W062835 | CGP77675 | Inhibitor | 99.46% | Unkown |
| HY-10330 | Toceranib | Inhibitor | 97.41% | Unkown |
| HY-144707 | AK-778-XXMU | 99.96% | Unkown | |
| HY-P1663 | ATWLPPR Peptide | Inhibitor | 99.63% | Unkown |
| HY-18302 | c-Kit-IN-5-1 | Inhibitor | 98.03% | Unkown |
| HY-W002616 | 5-Bromoindolin-2-one | 99.50% | Unkown | |
| HY-13838 | PLX647 | Inhibitor | 99.74% | Unkown |
| HY-15814 | HG-7-85-01 | 98.14% | Unkown | |
| HY-13785 | ZM 306416 | Inhibitor | 99.80% | Unkown |
| HY-P5438 | Srctide | Substrate | 99.71% | Unkown |
| HY-101219 | VEGFR-IN-1 | Inhibitor | 99.07% | Unkown |
| HY-125741 | GW768505A free base | Inhibitor | 99.26% | Unkown |
| HY-10517A | (Z)-Orantinib | Inhibitor | 99.44% | Unkown |
| HY-15769 | WHI-P180 | Inhibitor | 99.84% | Unkown |
| HY-132135 | (1E)-CFI-400437 dihydrochloride | Inhibitor | 98.08% | Unkown |
| HY-133551 | WF-47-JS03 | Inhibitor | 99.63% | Unkown |
| HY-119757 | Tyrphostin AG1433 | Inhibitor | 99.08% | Unkown |
| HY-RS07226 | KDR Human Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
| HY-148742 | RET-IN-21 | Inhibitor | 97.00% | Unkown |
| HY-RS07227 | Kdr Mouse Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
| HY-118105 | RK-20448 | Inhibitor | 99.38% | Unkown |
| HY-50751G | Linifanib (GMP) | Inhibitor | / | Unkown |
| HY-100824 | PP2 Analog | Inhibitor | / | Unkown |
| HY-10260S | Vandetanib-d6 | / | Unkown | |
| HY-10260S1 | Vandetanib-d4 | / | Unkown | |
| HY-10260S2 | Vandetanib-13C6 | / | Unkown | |
| HY-10330S | Toceranib-d8 | Inhibitor | 99.08% | Unkown |
| HY-116190 | CFI-401870 | Inhibitor | / | Unkown |
| HY-117733 | Zerumin A | Inhibitor | / | Unkown |
| HY-120214 | TAS05567 | Inhibitor | / | Unkown |
| HY-123586 | L-783277 | Inhibitor | / | Unkown |
| HY-13838A | PLX647 dihydrochloride | Inhibitor | / | Unkown |
| HY-146369 | PROTAC VEGFR-2 degrader-2 | Degrader | / | Unkown |
| HY-14979 | ML786 | Inhibitor | / | Unkown |
| HY-14979A | ML786 dihydrochloride | Inhibitor | / | Unkown |
| HY-15334 | CEP-5214 | Inhibitor | / | Unkown |
| HY-168114 | Multi-kinase inhibitor 3 | Inhibitor | / | Unkown |
| HY-168115 | Multi-kinase inhibitor 4 | Inhibitor | / | Unkown |
| HY-172487 | DSPE-PEG1000-K237 | / | Unkown | |
| HY-172488 | DSPE-PEG2000-K237 | / | Unkown | |
| HY-172488A | DSPE-PEG3400-K237 | / | Unkown | |
| HY-172489 | DSPE-PEG5000-K237 | / | Unkown | |
| HY-175477 | UNC9750 | Inhibitor | / | Unkown |
| HY-18318 | Takeda-6D | Inhibitor | 99.41% | Unkown |
| HY-18692 | Multi-kinase-IN-12 | Inhibitor | / | Unkown |
| HY-N16797 | Sanggenol C | / | Unkown | |
| HY-RS07228 | Kdr Rat Pre-designed siRNA Set A | Pre-designed Set | / | Unkown |
| HY-W062835A | CGP77675 hydrate | Inhibitor | / | Unkown |
| HY-W701071 | Vatalanib-d4 | / | Unkown | |
| HY-110045 | ZM-306416 hydrochloride | Inhibitor | / | Unkown |
| HY-119757A | Tyrphostin AG1433 hydrochloride | Inhibitor | / | Unkown |
| HY-149451 | SYHA1815 | Inhibitor | / | Unkown |
| HY-15769A | WHI-P180 hydrochloride | Inhibitor | / | Unkown |
| HY-174593 | Human KDR mRNA | / | Unkown | |
| HY-183616 | VEGFR-2-IN-87 | Inhibitor | / | Unkown |
| HY-N10379 | 19-epi-Scholaricine | 99.14% | Unkown | |
| HY-101628 | VEGFR-2-IN-9 | Inhibitor | / | Unkown |
Bioactive MoleculesInhibitory Antibodies
(6)
| Cat. No. | Product Name |
Effect
|
Purity |
Rare Diseases
|
|---|---|---|---|---|
| HY-P991141 | Inlecitug | Ligand | 98.62% | Unkown |
| HY-P991689 | Girancitug | Inhibitor | 98.80% | Unkown |
| HY-P990318 | Alacizumab | Inhibitor | / | Unkown |
| HY-P990542 | Anti-VEGFR2/KDR/CD309 Antibody | Inhibitor | / | Unkown |
| HY-P990543 | Anti-VEGFR2/KDR/CD309 Antibody (AT001) | Inhibitor | / | Unkown |
| HY-P991420 | UB-925 | Inhibitor | / | Unkown |